Lasinavir-CGP-61755-生命科学试剂-MCE.docxVIP

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Inhibitors?ScreeningLibraries?Proteins

www.MedChemE

Lasinavir

Cat.No.:HY-19260

CASNo.:175385-62-3

Synonyms:CGP61755;BMS-234475

分?式:C??H??N?O?

分?量:659.81

作?靶点:HIVProtease

作?通路:Anti-infection;MetabolicEnzyme/Protease

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性Lasinavir(CGP61755)

?种选择性HIV-1蛋?酶(HIV-1protease)抑制剂，其IC50值为1nM。Lasinavir可

?于HIV-1感染研究[1]。

IC50TargetIC50:1nM(HIV-1protease)[1]

REFERENCES

[1].CozensRM,etal.Synthesisandpharmacologicalevaluati