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VEGFR-2PathwayandFunctionEndothelialCellFlk-1/KDR
(VEGFR-2)Growth,Migration,
Permeability,Anti-apoptosisVEGFKinaseActivationCascadePPPLCVEGF-CVEGF-DAgentsTargetingVEGFR-2SignalinginDevelopmentAgentClassTargetAvastin?(bevacizumab)RecombinanthumanizedmonoclonalantibodyVEGF-AZD6474SmallmoleculeVEGFR-2SU-6668SmallmoleculeVEGFR-1,VEGFR-2,FGFR-1,andPDGFR-?PTK787SmallmoleculeVEGFR-1andVEGFR-2IMC-2C6FullyhumanmonoclonalantibodyVEGFR-2基因治疗基因治疗基因治疗基因治疗肿瘤靶向治疗与临床抗体-美罗华(Mabthera)03-12-22抗体-美罗华(Mabthera)第一个获准用于治疗人类肿瘤的单抗1997年11月美国FDA批准
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