有机合成讲义HETEROCYCLE1.pptVIP

Synthesis of heterocycles * I. Nomenclature of heterocycles 1. Five-membered heterocycles furan pyrrole thiophene 呋喃 吡咯 噻吩 imidazole 咪唑 pyrazole oxazole thiazole isoxazole isothiazole 吡唑 恶唑 噻唑 异恶唑 异噻唑 oxazoline thiazolidine 恶唑啉 噻唑烷 1,2,4-triazole 1,2,4-三唑 2. Six-membered heterocycles pyridine pyrimidine piperidine pyrazine 2H-pyran 4H-pyran pyridazine piperazine 1,2,4-triazine 1,3,5-triazine 吡啶 嘧啶 吡嗪 2H-吡喃 哌啶 哌嗪 哒嗪 三嗪 3. Fused heterocycles indole quinoline isoquinoline purine phenothiazine carbazole 吲哚 喹啉 异喹啉 嘌呤 吩噻嗪 咔唑 II. Synthesis of four-membered heterocycles 1. Cyclization 2. [ 2 + 2 ] C