执业药师药物化学习题集：抗生素与抗菌药物分类及结构.pdfVIP

Chapter1

Antibiotics

一、A

1.Whichofthefollowingdrugsdoesnothaveacidoralkalineproperties

A.Tetracycli

neB.

NorfloxacinC.

PenicillinGD.

DoxycyclineE.

Metacycline

2.Thereare3chiralcarbonatomsinthechemicalstructureofpenicillin,andtheirabsolute

configurationis

A.2R,5R,6R

B.2S,5S,6S

C.2S,5R,6R

D.2S,5S,6R

E.2S,5R,6S

3.Whichdrughasthefollowingchemicalstructure

A.Amtranan

B.Clavenic

acidC.

Temoxicillin

D.Adinicillin

E.Penicillin

G

4.Whichofthefollowingdrugsbelongstocarbapenemantibiotics

A.SubactamB.

ImipenemC.

ClavenicacidD.

Gentamicinsulfate

E.

Acetylspiromycin

5、哌拉西林属于哪一类抗菌药

A.大环内酯类

B.氨基糖苷类

C.β-内酰胺类

D.四环素类

E.其他类

6、第一个含氮的15元大环内酯药物是

A.琥乙红霉素

B.克拉霉素

C.罗红霉素

D.阿奇霉素

E.多西环素

7、阿米卡星的临床应用是

A.抗高血压药

B.抗菌药

C.抗疟药

D.

E.利尿药

8、下列各项哪一项符合头孢羟氨苄的特点

A.易溶于水

B.在体内可迅速代谢

C.不能口服

D.为口服的半合成头孢菌素

E.对耐药金葡萄球菌无作用

9、下列哪项与青霉素G性质不符

A.易产生耐药性

B.易发生过敏反应

C.可以口服给药

D.对革兰阳性菌效果好

E.为生物合成的抗生素

5.Whichantibacterialdrugispiperacillin

A.MacrolideB.

A

minoglycosides

C.β-lactamsD.

TetracyclinesE.

Othercategories

6.Thefirst15-membermacrolidedrugcontaining

nitrogenis

A.

Ethionomycin

B.ClarimycinC.

Ethionomycin

D.Azithro

mycinE.

Doxycycline

7.TheclinicalapplicationofAmikacinis

A.

Antihypertensive

drugsB.

Antibacterialdrugs

C.Antimalarial

drugsD.

AnestheticdrugsE.

Diureticdrugs

8.Whichofthefollowingitemsmeetsthecharacteristicsofcefoxoxyl

A.EasytosolubleinwaterB.Itcanbe

metabolizedquicklyinthebodyC.It

cannotbetakenorallyD.Itisa

semi-syntheticcephalosporinorallyE.It

hasnoeffectondrug-resistant

Staphylococcusaureus

9.Whichofthefollowingdoesnotmatchthe