- 1、原创力文档(book118)网站文档一经付费(服务费),不意味着购买了该文档的版权,仅供个人/单位学习、研究之用,不得用于商业用途,未经授权,严禁复制、发行、汇编、翻译或者网络传播等,侵权必究。。
- 2、本站所有内容均由合作方或网友上传,本站不对文档的完整性、权威性及其观点立场正确性做任何保证或承诺!文档内容仅供研究参考,付费前请自行鉴别。如您付费,意味着您自己接受本站规则且自行承担风险,本站不退款、不进行额外附加服务;查看《如何避免下载的几个坑》。如果您已付费下载过本站文档,您可以点击 这里二次下载。
- 3、如文档侵犯商业秘密、侵犯著作权、侵犯人身权等,请点击“版权申诉”(推荐),也可以打举报电话:400-050-0827(电话支持时间:9:00-18:30)。
- 4、该文档为VIP文档,如果想要下载,成为VIP会员后,下载免费。
- 5、成为VIP后,下载本文档将扣除1次下载权益。下载后,不支持退款、换文档。如有疑问请联系我们。
- 6、成为VIP后,您将拥有八大权益,权益包括:VIP文档下载权益、阅读免打扰、文档格式转换、高级专利检索、专属身份标志、高级客服、多端互通、版权登记。
- 7、VIP文档为合作方或网友上传,每下载1次, 网站将根据用户上传文档的质量评分、类型等,对文档贡献者给予高额补贴、流量扶持。如果你也想贡献VIP文档。上传文档
查看更多
Bioconjugate Chem. 2010, 21, 2213–2221 2213
Carborane-Conjugated 2-Quinolinecarboxamide Ligands of the
Translocator Protein for Boron Neutron Capture Therapy
Andrea Cappelli,*,† Salvatore Valenti,† Alessandra Mancini,† Germano Giuliani,† Maurizio Anzini,†
Saverio Altieri,‡,§ Silva Bortolussi,‡,§ Cinzia Ferrari,| Anna Maria Clerici,| Cecilia Zonta,| Fabio Carraro,⊥
Irene Filippi,⊥ Gianluca Giorgi,∇ Alessandro Donati,† Sandra Ristori,O Salvatore Vomero,† Alessandra Concas,# and
Giovanni Biggio#
Dipartimento Farmaco Chimico Tecnologico and European Research Centre for Drug Discovery and Development, Universita` degli
Studi di Siena, Via A. Moro, 53100 Siena, Italy, Dipartimento di Fisica Nucleare e Teorica, Universita` di Pavia, Via Ugo Bassi 6,
27100 Pavia, Italy, Istituto Nazionale di Fisica Nucleare (INFN), Sezione di Pavia, Via Ugo Bassi 6, 27100 Pavia, Italy, Dipartimento
di Scienze Chirurgiche, Laboratorio di Chirurgia Sperimentale, Universita` di Pavia, Via Ferrata 9, 27100 Pavia, Italy, Dipartimento di
Fisiologia, Universita` degli Studi di Siena, Via A. Moro, 53100 Siena, Italy, Dipartimento di Biologia Sperimentale “B. Loddo”,
Universita` degli Studi di Cagliari, Cittadella Universitaria, SS 554 (km 4.500), 09042 Monserrato (Cagliari), Italy, Dipartimento di
Chimica, Universita` di Siena, Via A. Moro, 53100 Siena, Italy, and Dipartimento di Chimica and CSGI, Universita` di Firenze, Via
della Lastruccia 7, 50019 Sesto Fiorentino, Italy. Received April 27, 2010; Revised Manuscript Received October 26, 2010
Potential boron neutron capture therapy (BNCT) agents have been designed on the basis of the evidence about
translocator protein (TSPO) overexpression on the outer mitochondrial membrane of tumor cells. The structure
of the first TSPO ligand bearing a carborane cage (compound 2d) has been
您可能关注的文档
- Chemistry Handouts Reduction化学讲义减少.pdf
- Knowledge based resource management for multifunction radar基于知识的多功能雷达资源管理.pdf
- Compendium Vol12 0289纲要.pdf
- Organometallic Chemistry b609350g有机金属化学.pdf
- Compendium Vol 纲要.pdf
- Catalytic Asymmetric Conjugate Addition催化不对称共轭加成反应.pdf
- Ag Mediated Reactions Coupling and Heterocyclization Reactions银介导的反应偶联反应和杂环化反应.pdf
- Materials Visualizer材料展示台.pdf
- Organometallic Chemistry b609347g有机金属化学.pdf
- Haake Rheomixe英文电子书r.pdf
- book Lecture notes on Logically Switched Dynamical systems关于逻辑交换动力学系统的讲义.pdf
- Pseudospin symmetry as a relativistic dynamical symmetry假旋光对称性作为相对论动力学对称性.pdf
- Compendium Vol12 0245纲要.pdf
- Compendium Vol12 0307简报.pdf
- Haunted Houses of New York City纽约市闹鬼的房子.pdf
- Electron Spin Resonance Spectroscopy电子自旋共振谱.pdf
- Thermoelectric performance of half Heusler compounds TiNiSn and TiCoSb半赫斯勒化合物和的热电性能.pdf
- Structural Information from Neutron Diffraction中子衍射的结构信息.pdf
- Living High and Letting Die高高在上让死亡.doc
- Cascade adaptive speed control of a thyristor driven DC motor晶闸管驱动直流电机的级联自适应速度控制.pdf
文档评论(0)