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Amdakefalin

Cat.No.:HY-109166

CASNo.:2253747-71-4

分⼦式:C₃₇H₅₃N₇O₆

分⼦量:691.86

Sequence:d-{Phe-Phe-Leu-Lys(3,6-Diazabicyclo[3.1.1]heptane-3-acetica

cid)}

SequenceShortening:d-{FFL-Lys(3,6-Diazabicyclo[3.1.1]heptane-3-aceticacid)}

作⽤靶点:OpioidReceptor

作⽤通路:GPCR/GProtein;NeuronalSignaling

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性Amdakefalin是⼀种μ和δ阿⽚受体(μ和δopioidreceptors)激动剂，具有镇痛作⽤。

IC50TargetμOpioidReceptor/MORδOpioidReceptor/DOR

REFERENCES

[1].WHODrugInformation,Vol.33,No.4,2019.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

Forresearchuseonly.

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