Fadaltran-BAY-1193397-生命科学试剂-MCE.pdfVIP

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Fadaltran

Cat.No.:HY-109130

CASNo.:1799809-36-1

Synonyms:BAY1193397

分⼦式:C₂₄H₂₉N₅O₂

分⼦量:419.52

作⽤靶点:AdrenergicReceptor

作⽤通路:GPCR/GProtein;NeuronalSignaling

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性Fadaltran(BAY1193397)是⼀种⼝服有效的α2C肾上腺素受体(α2C-adrenoreceptor)拮抗剂。Fadaltran

可⽤于糖尿病⾜溃疡的研究。

IC50TargetAlpha-2Cadrenergicreceptor

REFERENCES

[1].KapsaS,etal.Pharmacokinetics,Safety,andTolerabilityoftheα2C-AdrenoreceptorAntagonistBAY1193397inHealthyMale

Subjects.ClinPharmacolDrugDev.2022Mar;11(3):296-308.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

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