preparation of candesartan and atorvastatin nanoparticles by solvent evaporation坎地沙坦和阿托伐他汀的制备纳米粒子在溶剂蒸发.pdfVIP

preparation of candesartan and atorvastatin nanoparticles by solvent evaporation坎地沙坦和阿托伐他汀的制备纳米粒子在溶剂蒸发.pdf

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preparation of candesartan and atorvastatin nanoparticles by solvent evaporation坎地沙坦和阿托伐他汀的制备纳米粒子在溶剂蒸发

Molecules 2012, 17, 13221-13234; doi:10.3390/molecules171113221 OPEN ACCESS molecules ISSN 1420-3049 /journal/molecules Article Preparation of Candesartan and Atorvastatin Nanoparticles by Solvent Evaporation † Eliska Vaculikova 1,2,*, Veronika Grunwaldova 3,4, Vladimir Kral 3, Jiri Dohnal 1,5 and Josef Jampilek 1,5,* 1 Faculty of Pharmacy, University of Veterinary and Pharmaceutical Sciences, Palackeho 1/3, 612 42 Brno, Czech Republic 2 Nanotechnology Centre, VSB—Technical University of Ostrava, 17. listopadu 15/2172, 708 33 Ostrava, Czech Republic 3 Institute of Chemical Technology, Faculty of Chemical Engineering, Technicka 5, 166 28 Prague 6, Czech Republic 4 Institute of Inorganic Chemistry, Academy of Science, 250 68 Rez, Czech Republic 5 Research Institute for Pharmacy and Biochemistry, Lidicka 1879/48, 602 00 Brno, Czech Republic † Preliminary results were presented at The Sixteenth Electronic Conference on Synthetic Organic Chemistry (ECSOC-16, /presentation/1008), 1–30 November, 2012 (paper B1008). * Authors to whom correspondence should be addressed; E-Mails: eliskavaculikova@seznam.cz (E.V.); josef.jampilek@ (J.J.); Tel.: +420-541 -562-925 (J.J.); Fax: +420-541-240-607 (J.J.). Received: 8 October 2012; in revised form: 31 October 2012 / Accepted: 2 November 2012 / Published: 6 November 2012 Abstract: The solubility, absorption and distribution of a drug are involved in the basic aspects of oral bioavailability Solubility is an essential characteristic and influences the efficiency of

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