药学院2009年10共发表SCI论文9篇.docVIP

药学院2009年10月共发表SCI论文9篇 1、 标题：Convenient and versatile synthesis of formyl-substituted benzoxaboroles 作者: Ye L (Ye, Long)1, Ding DZ (Ding, Dazhong)1, Feng YQ (Feng, Yiqing)1, Xie DS (Xie, Dongsheng)1, Wu PH (Wu, Puhua)1, Guo H (Guo, Hui)1, Meng QQ (Meng, Qingqing)1, Zhou HC (Zhou, Huchen)1 来源出版物: TETRAHEDRON 卷: 65 期: 42 页: 8738-8744 出版年: OCT 17 2009 被引频次: 0 参考文献: 19 摘要: Despite of the medicinal significance of benzoxaboroles, with the newly discovered clinical compound AN2690 as an example, the synthetic method for rapid diversification of this novel scaffold is lacking. To this end, a versatile and scalable synthesis of formyl-substituted benzoxaboroles is described here. A key step is the mono-oxidation of the two hydroxyls in compound 4 by taking advantage of the stable oxaborole ring in non-coordinating solvents, which was devised based on the study of the intramolecular coordination and exchange properties. (C) 2009 Elsevier Ltd. All rights reserved. 文献类型: Article 语言: English KeyWords Plus: PINCER COMPLEXES; ANTIFUNGAL AGENT; ACID; DISCOVERY; DESIGN 通讯作者地址: Zhou, HC (通讯作者), Shanghai Jiao Tong Univ, Sch Pharm, 800 Dong Chuan Rd, Shanghai 200240, Peoples R China 地址: 1. Shanghai Jiao Tong Univ, Sch Pharm, Shanghai 200240, Peoples R China 电子邮件地址: hczhou@ 基金资助致谢: 基金资助机构 授权号 National Natural Science Foundation of China Shanghai Municipal Education Commission 07SG15 Science and Technology Commission of Shanghai Municipality 07pj14095 Ministry of Science and Technology of China 2009CB918404 Anacor Pharmaceuticals 出版商: PERGAMON-ELSEVIER SCIENCE LTD, THE BOULEVARD, LANGFORD LANE, KIDLINGTON, OXFORD OX5 1GB, ENGLAND 学科类别: Chemistry, Organic IDS 号: 504JE ISSN: 0040-4020 DOI: 10.1016/j.tet.2009.08.026 2、 标题：SYNTHESIS OF PYRROL[2,3-d]PYRIMIDINE ANALOGUES: PYRIDINE RING ANALOGUES OF PEMETREXED 作者: Xu Y (Xu, Yun)1, Yu MF (Yu, Mingfeng)1, Long Y (Long, Yan)1, Wu H (Wu, Han)1, Mao ZM (Mao, Zhenmin)1 来源出版物: HETE