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- 2026-01-30 发布于上海
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Fadolmidine
Cat.No.:HY-106388
CASNo.:189353-31-9
分⼦式:C₁₃H₁₄N₂O
分⼦量:214.26
作⽤靶点:AdrenergicReceptor
作⽤通路:GPCR/GProtein;NeuronalSignaling
储存⽅式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
⽣物活性Fadolmidine是⼀种选择性α2肾上腺素受体(α2-adrenoceptor)激动剂。Fadolmidine具有强效镇痛作⽤
,主要⽤于与脊髓⿇醉相关的疼痛控制研究[1]。
IC50Targetα2-adrenergicreceptor
REFERENCES
[1].LeinoT,etal.Effectsoffadolmidine,anα2‐adrenoceptoragonist,asanadjuvanttospinalbupivacaineonantinociceptionandmotorfunctionin
ratsanddogs[J].PharmacologyResearchPerspectives,2021,9(4):e00830.
McePdfHeight
Caution:Producthasnotbeenfullyvalidatedformedicalapplications.
Forresearchuseonly.
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