Ipazilide-fumarate-Win-54177-4-fumarate-生命科学试剂-MCE.pdfVIP

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Ipazilide-fumarate-Win-54177-4-fumarate-生命科学试剂-MCE.pdf

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Inhibitors•ScreeningLibraries•Proteins

www.MedChemE

Ipazilidefumarate

Cat.No.:HY-106330A

CASNo.:115436-74-3

Synonyms:Win54177-4fumarate

分⼦式:C₂₈H₃₄N₄O₅

分⼦量:506.59

作⽤靶点:PotassiumChannel

作⽤通路:MembraneTransporter/IonChannel

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性Ipazilidefumarate是⼀种抗⼼律失常剂。Ipazilidefumarate可降低K+去极化张⼒。Ipazilidefumarate可延

长⼼室不应期并具有抗异位搏动作⽤[1][2]。

REFERENCES

[1].GreenerY,etal.Chronic(1-year)safetyevaluationofipazilidefumarate,anantiarrhythmicagent,administeredorallytorats.Fundam

ApplToxicol.1993Feb;20(2):147-54.

[2].EzrinAM,etal.Invivoandinvitroeffectsofthenovelantiarrhythmicipazilideoncardiacandvascularsmoothmusclefunction[J].Drug

developmentresearch,1992,27(2):107-120.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

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