Moxidectin-Standard-CL301423-Standard-DataSheet-生命科学试剂-MCE.pdf

Moxidectin-Standard-CL301423-Standard-DataSheet-生命科学试剂-MCE.pdf

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Inhibitors•ScreeningLibraries•Proteins

www.MedChemE

Moxidectin(Standard)

Cat.No.:HY-B0777R

CASNo.:113507-06-5

Synonyms:CL301423(Standard)

分⼦式:C₃₇H₅₃NO₈

分⼦量:639.82

作⽤靶点:Antibiotic;BCRP;P-glycoprotein;Parasite

作⽤通路:Anti-infection;MembraneTransporter/IonChannel

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

溶解性数据

体外实验DMSO:100mg/mL(156.29mM;Needultrasonic)

H2O:0.1mg/mL(insoluble)

Mass

Solvent

1mg5mg10mg

Concentration

制备储备液1mM1.5629mL7.8147mL15.6294mL

5mM0.3126mL1.5629mL3.1259mL

10mM0.1563mL0.7815mL1.5629mL

BIOLOGICALACTIVITY

⽣物活性Moxidectin(Standard)是Moxidectin的分析标准品。本产品⽤于研究及分析应⽤。Moxidectin(CL301423)

是⼀种⼝服有效的⼤环内酯(ML)类驱⾍剂,可⽤于预防和控制⼼丝⾍和蛔⾍。Moxidectin在体内还是BCRP

和P-糖蛋⽩(P-gp)的底物,由Bcrp1和P-gp介导被分泌到母乳中,从宿主和寄⽣⾍中流出。这可能与⽜奶中

化合

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