Butriptyline-hydrochloride-Butriptylene-hydrochloride-生命科学试剂-MCE.pdfVIP

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Butriptyline-hydrochloride-Butriptylene-hydrochloride-生命科学试剂-MCE.pdf

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Inhibitors•ScreeningLibraries•Proteins

www.MedChemE

Butriptylinehydrochloride

Cat.No.:HY-A0175A

CASNo.:5585-73-9

Synonyms:Butriptylenehydrochloride

分⼦式:C₂₁H₂₈ClN

分⼦量:329.91

作⽤靶点:5-HTReceptor

作⽤通路:GPCR/GProtein;NeuronalSignaling

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性Butriptyline(Butriptylene)hydrochloride是⼀种具有⼝服活性的三环抗抑郁剂,可轻微增强中枢5-HT效应

。Butriptylinehydrochloride不抑制脑去甲肾上腺素摄取。Butriptylinehydrochloride可⽤于抑郁相关研究

[1][2][3]。

REFERENCES

[1].PugsleyTA,etal.Effectofbutriptylineonthebrainuptakemechanismsfornoradrenalineand5-hydroxytryptamine.JPharmPharmacol.

1974Oct;26(10):778-8.

[2].DullooAG,etal.Screeningofdrugsforthermogenicanti-obesityproperties:antidepressants.AnnNutrMetab.1987;31(2):69-80.

[3].MolinengoL,etal.Theactionofimipramine,amitriptyline,doxepinandbutriptylineinanoperantconditioningschedule.

Psychopharmacologia.1972;24(2):247-57.

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