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- 2026-02-06 发布于上海
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Inhibitors•ScreeningLibraries•Proteins
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NSD2-IN-5
Cat.No.:HY-177499
CASNo.:2604513-53-1
分⼦式:C₂₇H₂₅F₂N₉
分⼦量:513.54
作⽤靶点:HistoneMethyltransferase
作⽤通路:Epigenetics
储存⽅式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
⽣物活性NSD2-IN-5(Compound198)是NSD2抑制剂,IC50值介于0.001μM和0.01μM之间。NSD2-IN-5可⽤于
癌症研究。
IC50TargetNSD2
0.001-0.01μM(IC50)
REFERENCES
[1].HaibinDeng,etal.Piperidinyl-methyl-purineaminesasnsd2inhibitorsandanti-canceragents.WO2021026803A1.WIPO(PCT).2019-
08-14.
McePdfHeight
Caution:Producthasnotbeenfullyvalidatedformedicalapplications.
Forresearchuseonly.
Tel:400-820-3792;021Fax:021E-mail:tech@MedChemE
1/1MasterofBioactiveMolecules—您⾝边的抑制剂⼤师
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