AK-IN-1-DataSheet-生命科学试剂-MCE.pdf

Hotline: 400-820-3792 Inhibitors • Screening Libraries • Proteins www.MedChemE AK-IN-1 Cat. No.: HY-148327 CAS No.: 378775-98-5 分⼦式: C₂₂H₂₁N₃O₄ 分⼦量: 391.42 作⽤靶点: Adenosine Kinase 作⽤通路: Metabolic Enzyme/Protease; Neuronal Signaling 储存⽅式: Please store the product under the recommended conditions in the Certificate of Analysis. BIOLOGICAL ACTIVITY ⽣物活性 AK-IN-1 (化合物 4072-2732) 是⼀种对腺苷 (Ado) 有竞争性但对 ATP ⽆竞争性的腺苷激酶 (AK) 抑制剂。AK-IN- 1 浓度为 2, 4, 10 µM 时，能分别抑制 86%、87% 和 89% 的 AK 活性。AK-IN-1 在许多疾病领域 (包括缺⾎、炎 症和癫痫发作) 都具有较好的研究潜⼒。 REFERENCES [1]. Park J, et al. Identification and biochemical studies on novel non-nucleoside inhibitors of the enzyme adenosine kinase. Protein J. 2007 Apr;26(3):203-12. McePdfHeight Caution: Product has not been fully validated for medical applications. For research use only. Tel: 400-820-3792; 021 Fax: 021 E-mail: tech@MedChemE 1/1 Master of Bioactive Molecules — 您⾝边的抑制剂⼤师