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Inhibitors•ScreeningLibraries•Proteins
www.MedChemE
Octadecaneuropeptide
Cat.No.:HY-P11382
CASNo.:95237-86-8
Synonyms:ODN
分⼦式:C₈₁H₁₃₈N₂₄O₂₉
分⼦量:1912.11
Sequence:Gln-Ala-Thr-Val-Gly-Asp-Val-Asn-Thr-Asp-Arg-Pro-Gly-Leu-Le
u-Asp-Leu-Lys
SequenceShortening:QATVGDVNTDRPGLLDLK
作⽤靶点:GABAReceptor
作⽤通路:MembraneTransporter/IonChannel;NeuronalSignaling
储存⽅式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
⽣物活性Octadecaneuropeptide是⼀种由18个氨基酸残基组成的肽。Octadecaneuropeptide可衍⽣⾃Diazepam结
合抑制剂。Octadecaneuropeptide包含⼀个与γ-氨基丁酸受体调节位点(该位点通常被β-咔啉类物质占据)
特异性结合的配体。Octadecaneuropeptide能够以剂量依赖的⽅式增强惩罚引起的饮⽔抑制作⽤[1]。
REFERENCES
[1].FerreroP,etal.Studyofanoctadecaneuropeptidederivedfromdiazepambindinginhibitor(DBI):biologicalactivityandpresenceinrat
brain.ProcNatlAcadSciUSA.1986Feb;83(3):827-31.
McePdfHeight
Caution:Producthasnotbeenfullyvalidatedformedicalapplications.
Forresearchuseonly.
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