Octadecaneuropeptide-ODN-生命科学试剂-MCE.pdfVIP

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Inhibitors•ScreeningLibraries•Proteins

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Octadecaneuropeptide

Cat.No.:HY-P11382

CASNo.:95237-86-8

Synonyms:ODN

分⼦式:C₈₁H₁₃₈N₂₄O₂₉

分⼦量:1912.11

Sequence:Gln-Ala-Thr-Val-Gly-Asp-Val-Asn-Thr-Asp-Arg-Pro-Gly-Leu-Le

u-Asp-Leu-Lys

SequenceShortening:QATVGDVNTDRPGLLDLK

作⽤靶点:GABAReceptor

作⽤通路:MembraneTransporter/IonChannel;NeuronalSignaling

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性Octadecaneuropeptide是⼀种由18个氨基酸残基组成的肽。Octadecaneuropeptide可衍⽣⾃Diazepam结

合抑制剂。Octadecaneuropeptide包含⼀个与γ-氨基丁酸受体调节位点(该位点通常被β-咔啉类物质占据)

特异性结合的配体。Octadecaneuropeptide能够以剂量依赖的⽅式增强惩罚引起的饮⽔抑制作⽤[1]。

REFERENCES

[1].FerreroP,etal.Studyofanoctadecaneuropeptidederivedfromdiazepambindinginhibitor(DBI):biologicalactivityandpresenceinrat

brain.ProcNatlAcadSciUSA.1986Feb;83(3):827-31.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

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