NVS-PAK1-1-Standard-生命科学试剂-MCE.pdfVIP

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NVS-PAK1-1(Standard)

Cat.No.:HY-100519R

CASNo.:1783816-74-9

分⼦式:C₂₃H₂₅ClF₃N₅O

分⼦量:479.93

作⽤靶点:PAK;ReferenceStandards

作⽤通路:CellCycle/DNADamage;Cytoskeleton;Others

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性NVS-PAK1-1(Standard)是NVS-PAK1-1(HY-100519)的分析标准品。本产品⽤于研究及分析应⽤。NVS-

PAK1-1是⼀种化学探针，是有效，选择性的PAK1变构抑制剂，IC50值为5nM。

IC50TargetIC50:5nM(PAK1)[1]

REFERENCES

[1].KarpovAS,etal.OptimizationofaDibenzodiazepineHittoaPotentandSelectiveAllostericPAK1Inhibitor.ACSMedChemLett.2015

May22;6(7):776-81.

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Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

Forresearchuseonly.

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