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PHCCC(Standard)

Cat.No.:HY-100409R

CASNo.:179068-02-1

分⼦式:C₁₇H₁₄N₂O₃

分⼦量:294.31

作⽤靶点:mGluR;ReferenceStandards

作⽤通路:GPCR/GProtein;NeuronalSignaling;Others

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性PHCCC(Standard)是PHCCC(HY-100409)的分析标准品。本产品⽤于研究及分析应⽤。PHCCC是⼀种I型

mGluR(GroupImGluR)拮抗剂，IC50为3μM，PHCCC也是mGlu4受体选择性正向调节剂。具有抗帕⾦森

病作⽤。

REFERENCES

[1].MarinoMJetal.AllostericmodulationofgroupIIImetabotropicglutamatereceptor4:apotentialapproachtoParkinsonsdisease

treatment.ProcNatlAcadSciUSA.2003Nov11;100(23):13668-73.

[2].RécasensM,etal.Metabotropicglutamatereceptorsasdrugtargets.CurrDrugTargets.2007;8(5):651-681.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

Forresearchuseonly.

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